ChemInform Abstract: Straightforward and Facile Approach Toward the N‐Derivatization of Pyroglutamates Through Mitsunobu Reaction: Synthesis of N‐Alkyl/N‐Acyl Pyroglutamates.

Abstract

A simple and efficient methodology for the N‐alkylation/N‐acylation of pyroglutamate under Mitsunobu conditions is reported.