Erratum to “Synthesis and anticancer activity of 7-hydroxycoumarinyl gallates” [Pharmacol Rep 67 (2015) 236–244]

Hejchman, Elżbieta; Taciak, Przemysław; Kowalski, Sebastian; Maciejewska, Dorota; Czajkowska, Agnieszka; Borowska, Julia; Śladowski, Dariusz; Młynarczuk-Biały, Izabela

doi:10.1016/j.pharep.2015.05.015

Pharmacological Reports

2015

DOI: 10.1016/j.pharep.2015.05.015

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Erratum to “Synthesis and anticancer activity of 7-hydroxycoumarinyl gallates” [Pharmacol Rep 67 (2015) 236–244]

Elżbieta Hejchman

Przemysław Taciak

Sebastian Kowalski

et al.

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Cited by 2 publications

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“…The structures can serve as a base for creating new molecules with anticancer activity (9,10). Obtained compounds show high similarity with coumarin esters of gallic acid which appeared to have anticancer activity (10,11).…”

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Synthesis and anticancer activity evaluation of novel derivatives of 7-amino-4-methylquinolin-2(1H)-one

Kubica¹,

Taciak²,

Czajkowska³

et al. 2018

Acta Poloniae Pharmaceutica - Drug Research

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In this study, we designed and synthesized sixteen new derivatives of 7-amino-4-methylquinolin-2(1H)-one with potential anticancer activity. The structures of synthesized compounds were confirmed by 1H and 13 C NMR. The activity of novel substances was evaluated by cell viability assay and wound healing assay. In vitro tests for series of sixteen novel compounds were performed. The results showed that examined compounds are selective for a cancer cells, but their activity for various types of cancer is different. Three of the new compounds presented the ability to inhibit cells migration. The novel compounds constitute a good starting point for further studies and optimization of structure for new therapeutically effective anti-cancerous drugs. Seven compounds, which showed the highest rate of cell inhibition, were selected for further studies.

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confidence: 97%

Synthesis and anticancer activity evaluation of novel derivatives of 7-amino-4-methylquinolin-2(1H)-one

Kubica¹,

Taciak²,

Czajkowska³

et al. 2018

Acta Poloniae Pharmaceutica - Drug Research

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Synthesis and Antidepressant Evaluation of Heteroaromatic derivatives of Gallic Acid

Chaurasia,

Mishra,

Mishra

2023

RJPT

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Oxidative stress is a causative factor of depression and several studies have reported that gallic acid or the derivatives thereof had proven to be effective in displaying antidepressant like action in animal models. Owing to the antioxidant property of GA and the study of structural features it was hypothesized to design new small molecule antidepressant drugs based on GA containing piperazine/piperidine. The two step reaction involved the formation of acid chloride of GA and its conversion to the target compounds in presence of acetone. All the compounds were subjected to evaluation of antidepressant effect using the widely used TST and FST models in mice at dose of 40mg/kg intraperitoneally. The synthesized compounds 2b, 2c and 2e were able to reduce the immobility time in both the models as comparable to the reference compound fluoxetine (10mg/kg) while compounds 2a and 2d were not very significant in reducing the immobility of mice.

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Erratum to “Synthesis and anticancer activity of 7-hydroxycoumarinyl gallates” [Pharmacol Rep 67 (2015) 236–244]

Cited by 2 publications

References 0 publications

Synthesis and anticancer activity evaluation of novel derivatives of 7-amino-4-methylquinolin-2(1H)-one

Synthesis and anticancer activity evaluation of novel derivatives of 7-amino-4-methylquinolin-2(1H)-one

Synthesis and Antidepressant Evaluation of Heteroaromatic derivatives of Gallic Acid

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