CH Activation of Indolines, Tetrahydroquinolines, and Tetrahydroisoquinolines

Abstract

Indolines could be successfully applied in the diversity of CH bond functionalization of benzenoid moiety without the competition between sp 3 H and sp 2 H activations thereby offering an access to functionalized heterocycles including the indoles. The metal‐catalyzed transformations proceeding the CH functionalizations of C4, C5, C6, and C7 position will be covered in the article along with applications to analogs systems in tetrahydroquinolines and tetrahydroisoquinolines.