“…All these compounds are of biochemical and pharmacological interest as natural polyamine analogs. [14][15][16] The reported synthetic method for N-benzoyl-N 0 -aryl pentamethylenediamines involves the reaction of N-acylpiperidines with PCl 5 followed by aminolysis. 17 The overall yields are moderate, and the procedure is restricted to N-acyl derivatives without a-hydrogens.…”