ChemInform Abstract: Asymmetric Synthesis of Amino Acids by Enantio‐ and Diastereodifferentiating Reactions

Synthesis of New Racemic α,α-Diaminocarboxylic Ester Derivatives

“…The synthesis of amino acids was a very important development [ 7 ]. Their applications can be found currently in several domains: biochemistry, enzymology [ 8 , 9 , 10 , 11 ], medicine (antibiotics, antiepileptics, antivirals, antiprotozoals, cardiovascular, atherosclerosis, renal failure and diabetes, neuroexciters [ 12 , 13 , 14 , 15 , 16 , 17 , 18 , 19 , 20 , 21 , 22 , 23 , 24 , 25 , 26 ]), agrochemical industry (herbicides, fungicides, regulation of plant growth), in addition to their important utility as chiral auxiliaries in asymmetric synthesis [ 27 , 28 ].…”

Synthesis and Characterization of New Racemic α-Heterocyclic α,α-Diaminoester and α,α-Diamino Acid Carboxylic: 2-Benzamido-2-[(Tetrahydro-Furan-2-Ylmethyl)Amino]Acetate and 2-Benzamido-2-[(Tetrahydro-Furan-2-Ylmethyl)Amino] Acetic Acid

“…Given the very broad activity they present, research teams are interested in evaluating and developing their role for very effective use [1][2][3][4][5]. This has led to the development of numerous synthetic methods for a variety of compounds [6]. Heterocyclic chemistry is the basis for the discovery of the importance of the multiple medical properties of these compounds [7][8][9][10][11][12].…”

Synthesis of?-triazolyl?-amino acid derivatives

“…This has led to the development of numerous synthetic methods for a variety of compounds (Haemers et al, 1989;Williams, 1989). However the synthesis of heterocyclic amino acids has not been very well investigated to date.…”