2014
DOI: 10.1002/chin.201445127
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ChemInform Abstract: Palladium on Carbon‐Catalyzed One‐Pot N‐Arylindole Synthesis: Intramolecular Aromatic Amination, Aromatization, and Intermolecular Aromatic Amination.

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Cited by 2 publications
(2 citation statements)
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“…The two-step one-pot procedure for the preparation of N -arylindoles relies on the palladium-catalyzed cyclization of 2-bromophenethylamines S17-1 , which is followed by the palladium-catalyzed N -arylation of the resulting indoles S17-2a ( Scheme 17 ) [ 74 ]. The optimization of the reaction conditions revealed that the cyclization of amines S17-1 into indoles S17-3 must be carried out at 200 °C.…”
Section: Transition-metal-catalyzed N -Arylation Of Indolesmentioning
confidence: 99%
“…The two-step one-pot procedure for the preparation of N -arylindoles relies on the palladium-catalyzed cyclization of 2-bromophenethylamines S17-1 , which is followed by the palladium-catalyzed N -arylation of the resulting indoles S17-2a ( Scheme 17 ) [ 74 ]. The optimization of the reaction conditions revealed that the cyclization of amines S17-1 into indoles S17-3 must be carried out at 200 °C.…”
Section: Transition-metal-catalyzed N -Arylation Of Indolesmentioning
confidence: 99%
“…We recently disclosed the direct C-2 arylation of indoles in Trp-containing peptidic sequences in an intermolecular manner, without additional requierements 37 . Although the alternative N -arylation processes are conceivable, such Ullmann-type reactions take place normally with Cu and Pd catalysts, in the latter case usually requiring strong bases 40 . No experimental evidence of these transformations have been recorded in our systems.…”
mentioning
confidence: 99%