Abstract:The direct N-arylation of
cyclic amides can be considered a pivotal issue for modern organic chemistry.
Here, we report the method for copper-catalyzed <i>N</i>-arylation of diverse oxadiazolones by diaryliodonium salts in mild conditions in high
yields (up to 92%) using available CuI as a catalyst. The developed method
allows to efficiently utilize both symmetric and unsymmetric diaryliodonium
salts bearing auxiliary groups such as 2,4,6-trimethoxyphenyl (TMP). The evaluation
of steric effects in … Show more
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