2020
DOI: 10.1021/acsomega.0c01769
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Crystal Growth, Single Crystal Structure, and Biological Activity of Thiazolo-Pyridine Dicarboxylic Acid Derivatives

Abstract: Four novel TPDCA derivatives were prepared via a supersaturation method combining TPDCA with water, N-methyl-2-pyrrolidone (NMP), Na­(PO2H2), and ammonia solution: 2­(C9H7NO5S)­H2O (1), (C9H7NO5S)­C5H9NO (2), (C9H7NO5S)­Na­(PO2H2) (3), and (C9H5NO5S)­(NH4)2(H2O) (4). Their crystal structures were determined by single-crystal X-ray diffraction. Compounds (1) and (2) crystallize in the monoclinic space groups P21 and P21/c, respectively, whereas compounds (3) and (4) crystallize in the triclinic space group P1̅.… Show more

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Cited by 7 publications
(3 citation statements)
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“…Organic phosphates are highly lustrous, adherent, and ductile, and their additives are used in electroplating baths. Structure, as well as biological activities of thiazolo-pyridine dicarboxylic derivatives, were reported by Yahia et al [3]. Linear, as well as nonlinear optical properties of pyridine N-oxide, were reported by Soscun et al [4].…”
Section: Introductionmentioning
confidence: 87%
“…Organic phosphates are highly lustrous, adherent, and ductile, and their additives are used in electroplating baths. Structure, as well as biological activities of thiazolo-pyridine dicarboxylic derivatives, were reported by Yahia et al [3]. Linear, as well as nonlinear optical properties of pyridine N-oxide, were reported by Soscun et al [4].…”
Section: Introductionmentioning
confidence: 87%
“…Antibacterial (against both gram-positive and gram-negative bacteria), antiviral, antifungal, antituberculose, and antiparasitic activity of compounds containing thiazolopyridine structure were reported [247][248][249][250][251]. Additionally, cytotoxic and anticancer activity of thiazolopyridine derivatives were investigated in many studies [252][253][254][255]. Moreover, there are many thiazolopyridine-bearing compounds with various bioactivity profile, such as histamine H3-receptor antagonistic activity, mGluR5metabotropic glutamate receptor subtype 5-antagonist, sphingosine-1-phosphate (S1P) agonist, DNA Gyrase B (GyrB) ATPase inhibitor, anti-inflammatory activity, phosphoinositide 3-kinase inhibitor, and allosteric inhibitor of MALT1 [129,[256][257][258][259][260][261].…”
Section: Thiazolopyridines and Isothiazolopyridinesmentioning
confidence: 99%
“…Antibacterial (against both gram-positive and gram-negative bacteria), antiviral, antifungal, antituberculose, and antiparasitic activity of compounds containing thiazolopyridine structure were reported [247][248][249][250][251]. Additionally, cytotoxic and anticancer activity of thiazolopyridine derivatives were investigated in many studies [252][253][254][255]. Exploring Chemistry with Pyridine Derivatives 132 Moreover, there are many thiazolopyridine-bearing compounds with various bioactivity profile, such as histamine H3-receptor antagonistic activity, mGluR5metabotropic glutamate receptor subtype 5-antagonist, sphingosine-1-phosphate (S1P) agonist, DNA Gyrase B (GyrB) ATPase inhibitor, anti-inflammatory activity, phosphoinositide 3-kinase inhibitor, and allosteric inhibitor of MALT1 [129,[256][257][258][259][260][261].…”
Section: Thiazolopyridines and Isothiazolopyridinesmentioning
confidence: 99%