2017
DOI: 10.1002/bkcs.11088
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Microwave‐assisted Solid‐phase Synthesis of N‐substituted‐2‐aminobenzo[d][1,3] Thiazine Derivatives from a BOMBA Resin

Abstract: An efficient solid‐phase methodology has been developed for the synthesis of N‐acyl and N‐sulfonyl substituted 2‐aminobenzo[d][1,3]thiazine derivatives. The key step in this methodology is the preparation of backbone amide linker‐bound 2‐aminobenzo[d][1,3]thiazine resin through cyclization reaction between isothiocyanates and BOMBA resin under microwave irradiation. This 2‐aminobenzo[d][1,3]thiazine core skeleton resin undergoes substitution reactions with various electrophiles, such as acid halides and sulfon… Show more

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Cited by 5 publications
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