Studies on Chemotherapeutics for Mycobacterium tuberculosis. XVIII. : Synthesis and Antibacterial Activity on Mycobacterium tuberculosis of Formyl-8-hydroxyquinoline Derivatives

Fujikawa, Fukujiro; Hirai, Kunio; Toyota, Takeshi; Tamada, Ryusuke; Kijun, Sai; Naito, Masukazu; Tsukuma, Shunji

doi:10.1248/yakushi1947.87.7_844

Cited by 5 publications

(2 citation statements)

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“…Among the class of hydroxyquinolines, the chemistry of 8-hydroxyquinolines (8HQs) has attracted special interest due to their diverse biological properties [1,2] such as antiamebic, [3] antiseptic and disinfectant, [4,5] antimalarial, [6] antituberculotic, [7] antidiuretic, [8] anticancer, [9,10] antibacterial and antifungal. [11 -13] 8HQ shows remarkable effects similar to the antibiotic, lomofugin, which rapidly and selectively inhibits the RNA synthesis in yeast.…”

Section: Introductionmentioning

confidence: 99%

Synthesis and antimicrobial activities of sulfonohydrazide‐substituted 8‐hydroxyquinoline derivative and its oxinates

Dixit¹,

Vanparia²,

Patel³

et al. 2010

Applied Organom Chemis

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Section: Introductionmentioning

confidence: 99%

Synthesis and antimicrobial activities of sulfonohydrazide‐substituted 8‐hydroxyquinoline derivative and its oxinates

Dixit¹,

Vanparia²,

Patel³

et al. 2010

Applied Organom Chemis

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“…A number of biologically relevant entities containing the 1,3,4‐oxadiazole motif are used as HIV integrase inhibitors and angiogenesis inhibitors 13, 14. Among the class of hydroxyquinolines, the chemistry of 8‐hydroxyquinolines has attracted special interest due to their diverse biological properties15, 16 such as antiamebic,17 antiseptic and disinfectant,18, 19 antimalarial,20 antituberculotic,21 antidiuretic,22 anticancer,23, 24 antibacterial and antifungal 25, 26. 5‐Chlromethyl‐8‐quinolinol (CMQ) can be synthesized easily and studied extensively 27.…”

Section: Introductionmentioning

confidence: 99%

Antibacterial, spectral and thermal aspects of some novel first transition metal‐based heterochelates

Oza

Jani

Patel

2010

Applied Organom Chemis

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1 H NMR, 13 C NMR and IR spectroscopic techniques and reacted with transition metal salts to afford metalcontaining heterochelates. The structures of the synthesized heterochelates were characterized using elemental analyses, infrared spectra, electronic spectra, magnetic measurements, FAB mass spectrum and thermogravimetric analyses. The kinetic parameters such as order of reaction (n) and the energy of activation (E a ) are reported using the Freeman-Carroll method. The pre-exponential factor (A), the activation entropy ( S # ), the activation enthalpy ( H # ) and the free energy of activation ( G # ) were calculated. Heterochelates were also screened for their in vitro antibacterial activity against a range of Gram-positive (Bacillus substilis, Staphylococcus aureus) and Gram-negative (Escherichia coli, Serratiamarcescens) organisms.

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Quinoline Aldehydes

Greenhill¹

1990

Chemistry of Heterocyclic Compounds: A Series of Monographs

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Studies on Chemotherapeutics for Mycobacterium tuberculosis. XVIII. : Synthesis and Antibacterial Activity on Mycobacterium tuberculosis of Formyl-8-hydroxyquinoline Derivatives

Cited by 5 publications

References 0 publications

Synthesis and antimicrobial activities of sulfonohydrazide‐substituted 8‐hydroxyquinoline derivative and its oxinates

Synthesis and antimicrobial activities of sulfonohydrazide‐substituted 8‐hydroxyquinoline derivative and its oxinates

Antibacterial, spectral and thermal aspects of some novel first transition metal‐based heterochelates

Quinoline Aldehydes

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