Synthesis and characterization of technetium(V) complexes with N-(thiocarbamoyl)benzamidines. X-ray crystal structure of bis[N-(N,N-diethylthiocarbamoyl)benzamidinato]oxotechnetium(V) chloride, [TcO(et2tcb)2]Cl

Aqueous solubilities of five N-(diethylaminothiocarbonyl)benzimido derivatives at T = 298.15 K

“…They are accessible through the reaction of coordinated N-Acylthiourea with acid chlorides, followed by further derivatisation. Members of this family are known chelating agents (Hartung et al, 1985), with potential applications e.g., radio pharmaceuticals ( 99m Tc) (Abram et al, 1989). A large number of serine proteinase inhibitors has been developed, starting from benzamidine and its derivatives (Ensinck et al, 1972;Henkel et al, 1983;Jeffcoate and White, 1974).…”

Thermochemical studies of two N-(diethylaminothiocarbonyl)benzimido derivatives

“…These compounds have been investigated due to their application as radiopharmaceuticals ( 99m Tc) [3]. Benzamidines and a variety of their derivatives are known starting materials for a large number of Serine proteinase inhibitors [4][5][6].…”

Thermochemical studies of three N-thiocarbamoylbenzamidines

“…These compounds have been investigated due to their application as radio pharmaceuticals ( 99m Tc) [3]. It is also a very well-known fact that a large number of serine proteinase inhibitors has been developed, starting from benzamidine and its derivatives [4][5][6].…”