In this study, we present new U–Pb zircon ages and whole‐rock major and trace element data for the late Carboniferous–Middle Jurassic intrusive rocks in the Helong area, NE China. These data constrain the timing of tectonic transition from the Paleo‐Asian oceanic regime to the circum‐Pacific regime. U–Pb zircon dating indicates that the late Carboniferous–Middle Jurassic magmatic events in the Helong area can be subdivided into late Carboniferous, middle Permian, Early–Middle Triassic, Late Triassic, Early Jurassic, and early Middle Jurassic. The late Carboniferous granodiorites and middle Permian monzogranites belong to the calc‐alkaline series and have an affinity to I‐type granitoids, suggesting that they formed in a typical Andean‐type continental arc setting due to the southward subduction of the Paleo‐Asian oceanic plate beneath the NCC. The Middle Triassic granodiorites and monzogranites in the Helong area exhibit an affinity to adakitic rocks with their parental magma derived by the partial melting of thickened lower continental crust. The Late Triassic I‐type monzogranites and coeval ultramafic–mafic rocks constitute a bimodal igneous rock association, together with coeval A‐type granites and rhyolites, signifying an extensional environment. Combined with the absence of 240‐ to 225‐Ma sedimentation, the study area experienced a change from Early–Middle Triassic compression to Late Triassic extension related to the final closure of the Paleo‐Asian Ocean. The Early–early Middle Jurassic gabbros, diorites, granodiorites, and monzogranites are calc‐alkaline in nature and enriched in LREE and LILE but depleted in HREE and HFSE. Combined with the spatial variations in K contents of Early Jurassic igneous rocks in NE China from the continental margin to intracontinental region, and the presence of an Early Jurassic accretionary complex, we suggest that Early–early Middle Jurassic magmatism in the Helong area formed in an active continental margin setting related to the subduction of the Paleo‐Pacific Plate beneath Eurasia. We conclude that the tectonic transition from the Paleo‐Asian oceanic regime to the circum‐Pacific regime occurred in the Late Triassic–Early Jurassic.