The Synthesis and Vasopressin (AVP) Antagonist Activity of a Novel Series of N- 4,5,thieno [3,2b]azepines.-Fifteen compounds of type (XI) are prepared and tested along with four known compounds of similar structure as arginine vasopressin (AVP) receptor antagonists. It is shown that enhanced in vivo (po) activity is found when the 2-phenylbenzoyl substituent is present in the molecule, cf. (XIb). -(ALBRIGHT, J. DONALD; DELOS SANTOS, EFREN G.; DUSZA, JOHN P.; CHAN, PETER S.; COUPET, JOSEPH; RU, XUN; MAZANDARANI, H.; Bioorg. Med.
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