A series of cationic gold(I) complexes containing 1-[2-(acridin-9-ylamino)ethyl]-1,3-dimethylthiourea (1), [AuL(1)]n+ (where L is Cl−, Br-, SCN−, PEt3, PPh3, or 1), derived from a class of analogous platinum(II) antitumor agents, has been synthesized. Unlike platinum, gold does not form permanent adducts with DNA, and its complexes are two orders of magnitude less cytotoxic in non-small-cell lung cancer cells than the most active platinum-based agent. Instead, several gold analogues show submicromolar and selective antimicrobial activity against Mycobacterium tuberculosis.

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The seasonal variation in the chemical composition of the leaf essential oil of Zanthoxylum clava-herculis has been analyzed by GC-MS. Three individual trees were sampled four times during the course of the 2004 growing season. Notable differences were recorded in the essential oil yields from the three trees on the four collection dates; yields were highest in May and lowest in July The leaf essential oils were made up of 25 components, largely menthane monoterpenoids, dominated by limonene (44-73%) and 1,8-cineole (16-43%), with lesser amounts of α-thujene, linalool, γ-terpinene, and α-terpineol. The ratio of oxygenated monoterpenoids to monoterpene hydrocarbons generally increased during the season, largely reflected in the 1,8-cineole/limonene ratio.

The leaf oil of Calyptranthes pallens was obtained by hydrodistillation and analyzed by GC/MS. The most abundant oil components were the monoterpenoids α-pinene (24.7%), α-terpineol (13.8%), and trans-pinocarveol (11.6%). The antimicrobial activity against Bacillus cereus, Staphylococcus aureus, Escherichia coli, Pseudomonas aeruginosa, Candida albicans, and Aspergillus niger, and the in-vitro cytotoxicity of the oil on Hep G2, MDA-MB-231, Hs 578T, and PC-3 human tumor cells were also examined.