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Beckmann rearrangement was used as a key step to synthesize six-membered lactams fused to a heteroaromatic or aromatic system. Derivatives of biologically active scaffolds like β-and γ-carbolinone, dihydropyrrolopyridinone and tetrahydroisoquinolinone were synthesized using this strategy.

Indole derivatives R 0140Thermal and Microwave-Assisted Conjugate Additions of Indole on Electron--Deficient Nitro-Olefins. -The microwave-assisted conjugate addition of indole (I) to electron-deficient nitro-olefins (II) leads to significantly higher yields and proceeds much faster compared to classical methods such as heating in a sealed tube or via Grignard reaction. -(KUSURKAR*, R. S.; ALKOBATI, N. A. H.; GOKULE, A. S.; CHAUDHARI, P. M.; WAGHCHAURE, P. B.; Synth. Commun. 36 (2006) 7-9, 1075-1081; Dep. Chem., Univ. Pune, Pune 411 007, India; Eng.) -H. Haber 35-111

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