Diphenyl carbonate mediated synthesis of amides of carboxylic acids: Facile synthesis of drug molecules and drug intermediates

Prachi, Ramteke; Gill, Manjinder Singh

doi:10.1016/j.tetlet.2023.154621

Tetrahedron Letters

2023

DOI: 10.1016/j.tetlet.2023.154621

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Diphenyl carbonate mediated synthesis of amides of carboxylic acids: Facile synthesis of drug molecules and drug intermediates

Ramteke Prachi,

Manjinder Singh Gill

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2024

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Cited by 4 publications

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Recent Advances in Direct Amidation Via Organocatalysis

Hussein,

Hassoon Mageed

2024

Asian J Org Chem

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The formation of amide bonds is essential for a wide range of applications in biological and organic systems, including proteins, pesticides, polymers, and pharmaceuticals. Moreover, it plays a critical role in the synthesis of numerous bioactive compounds with anticancer, antibacterial, and antifungal properties. Due to the limitations of conventional coupling reagents for amide synthesis, there is a growing demand for environmentally sustainable methodologies, particularly the direct formation of amides from carboxylic acids and amines. Over recent years, we have developed several catalytic reactions based on organocatalysis, advancing sustainable synthetic methods in both organic and medicinal chemistry. This review comprehensively discusses catalytic amidation reactions published up to January 2024, focusing on both organocatalysis and boron‐based catalysis for the direct condensation of carboxylic acids and amines. Additionally, it highlights our recent contributions to sustainable amidation protocols, which are progressively replacing traditional catalytic approaches in modern synthetic chemistry.

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Recent Advances in Direct Amidation Via Organocatalysis

Hussein,

Hassoon Mageed

2024

Asian J Org Chem

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Discovery of novel osthole derivatives exerting anti-inflammatory effect on DSS-induced ulcerative colitis and LPS-induced acute lung injury in mice

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et al. 2024

European Journal of Medicinal Chemistry

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Development of new dehydrocostuslactone derivatives for treatment of atopic dermatitis via inhibition of the NF-κB signaling pathway

Li,

Lu,

et al. 2024

RSC Med. Chem.

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Diphenyl carbonate mediated synthesis of amides of carboxylic acids: Facile synthesis of drug molecules and drug intermediates

Cited by 4 publications

References 50 publications

Recent Advances in Direct Amidation Via Organocatalysis

Recent Advances in Direct Amidation Via Organocatalysis

Discovery of novel osthole derivatives exerting anti-inflammatory effect on DSS-induced ulcerative colitis and LPS-induced acute lung injury in mice

Development of new dehydrocostuslactone derivatives for treatment of atopic dermatitis via inhibition of the NF-κB signaling pathway

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