New Efficient Synthesis of 3-Carboxylquinolines

Abstract

ABSTRACT. Rapid and efficient synthesis of substituted 3-carboxylquinoline derivatives from 4-chloro-3-formylcoumarin and substituted anilines using 30% H2SO4 in methanol at room temperature within the duration of 5-30 min., through domino condensation-cyclization-ring opening reaction.

Antibacterial Screening of some Heterocyclic Compounds Containing Quinoline Nucleus

“…These derivatives are also used for the preparation of nano-and meso structures having enhanced electronic and photonic properties [9,10] and are known to have applications as pharmaceuticals, agrochemicals and synthetic building blocks [11]. Quinolines have been found to possess antimalarial, anti-bacterial, antifungal, antihelmintic, cardiotonic, anticonvulsant, anti-inflammatory, and analgesic activity [12][13][14][15][16][17][18].…”

Antibacterial Screening of some Heterocyclic Compounds Containing Quinoline Nucleus

“…These derivatives are also used for the preparation of nano-and meso structures having enhanced electronic and photonic properties [9,10] and are known to have applications as pharmaceuticals, agrochemicals and synthetic building blocks [11]. Quinolines have been found to possess antimalarial, anti-bacterial, antifungal, antihelmintic, cardiotonic, anticonvulsant, anti-inflammatory, and analgesic activity [12][13][14][15][16][17][18].…”