2014
DOI: 10.1016/j.jscs.2011.05.019
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Synthesis and in vitro antibacterial activity of new oxoethylthio-1,3,4-oxadiazole derivatives

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Cited by 26 publications
(18 citation statements)
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“…The first site is the sulfonamide group (─SO 2 NH─) which acts as an antimetabolite and competes with p ‐aminobenzoic acid for incorporation into folic acid. Thus, bacterial growth is limited through folate deficiency without effect on human cells …”
Section: Resultsmentioning
confidence: 99%
“…The first site is the sulfonamide group (─SO 2 NH─) which acts as an antimetabolite and competes with p ‐aminobenzoic acid for incorporation into folic acid. Thus, bacterial growth is limited through folate deficiency without effect on human cells …”
Section: Resultsmentioning
confidence: 99%
“…A series of 2(4‐pyridyl)‐5[(aryl/heteroarylamino)‐1‐oxoethyl]thio‐1,3,4‐oxadiazoles were synthesized by Ravel et al., resulting in identification of compounds 135 – 137 that caused more than 90% inhibition of M. tuberculosis at low concentrations ranged between 0.0052 and 0.0089 μM (Fig. ) …”
Section: Oxadiazolesmentioning
confidence: 99%
“…1,2 Due to their structural diversity their biological activities include antibacterial, 3,4 antitubercular, antifungal, cytotoxic, anticancer, 5,6 and many others. So far, our work has been based on the synthesis of 1,3,4-oxadiazoles, which are present in some well-known drugs like Furamizole (antibiotic), Raltegravir (antiretroviral), Zibotentan (anticancer), and tiodazosin and nesapidil (antihypertensive).…”
Section: Introductionmentioning
confidence: 99%