ChemInform Abstract: Synthesis of Acylthiosulfanilic Esters.

Lubenets, V. І.; Yarish, M. E.; Vid, L. V.; Chuiko, L.S.; Solonin, V. N.; Kucherenko, L. A.

doi:10.1002/chin.198723133

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2023

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“…The target esters of 4-methacryloylaminobenzenethiosulfonic acid (M5-M7) were obtained via acylation of the corresponding esters of 4-aminobenzenethiosulfonic acid with methacryloyl chloride, analogously to the procedure of obtaining 4'-methoxyphenyl and 4'nitrophenyl esters of 4-methacryloylaminobenzenethiosulfonic acid. 36…”

Section: Resultsmentioning

confidence: 99%

Obtaining and Determining Antiviral and Antibacterial Activity of S-Esters of 4-R-Aminobenzenethiosulfonic Acid

Zaczyńska¹,

Czarny²,

Карпенко³

et al. 2023

ChChT

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A number of S-esters of 4-R-aminobenzene¬thiosulfonic acids were synthesized via alkylation of the sodium salt of 4-acetylaminobenzenethiosulfonic acid with various alkylating agents and acylation of the corresponding esters of 4-aminobenzenethiosulfonic acid with metha-cryloyl chloride. For obtaining S-methyl 4-(acetyla-mino)benzenesulfonothioate, it was developed a synthetic technique corresponding to the basic principles of "green chemistry". The degree of compound cytotox-icity was measured by determining A-549 cell growth using colorimetric method. The antibacterial activity of the thiosulfonates was determined by the agar diffusion test and the antiviral action by their cytopathic effect at TCID50 value.

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Section: Resultsmentioning

confidence: 99%