Synthesis and in vivo nematocidal evaluation of novel 3-(trifluoromethyl)-1H-pyrazole-4-carboxamide derivatives

Synthesis and Insecticidal Activity of New Quinoline Derivatives Containing Perfluoropropanyl Moiety

“…In our previous work , we found that the perfluoropropanyl group on the quinoline ring can increase the fungicidal activity, so in line with our continued efforts to synthesize novel lead compounds for drug discover , the fungicide tebufloquin was selected as a lead compound, the t ‐Bu group was replaced by perfluoropropanyl group, the methyl group was replaced by chlorine atom, the fluorine atom was replaced by methyl group, and the ether group was replaced by ester carbonate. Our original strategy is depicted in Scheme .…”

Synthesis and in vivo fungicidal activity of some new quinoline derivatives against rice blast

“…The fluorine atom with a small radius and strong electronegativity has simulation, electronic, blocking, and penetration effects. Fluorine atoms are frequently introduced into herterocycles to obtain strong bioactivity in medicinal chemistry and pesticide chemistry.…”

Synthesis, crystal structure, and optical properties of fluorinated poly(pyrazole) ligands andin silicoassessment of their affinity for volatile organic compounds

“…Pyrazole and its derivatives have been extensively studied for their wide biological activities, [1][2][3] including antibacterial, 4 antifungal, [5][6][7][8] and insecticidal [9][10][11] properties. Furthermore, pyrazoles have been intensively employed as nitrogen-donor ligands in coordination chemistry.…”