Synthesis of 1,3-thiazine derivatives and their evaluation as potential antimycobacterial agents

Selenium‐Containing Heterocycles from Isoselenocyanates: Synthesis of 1H‐5‐Selena‐1,3,6‐triazaaceanthrylene Derivatives

“…[6][7][8][9][10]). For example, some organo-selenium compounds are active as insecticides and microbicides [11], as prooxidants [12], and antimycobacterial agents [13]. Recently, the research group of Koketsu published some novel syntheses of selenaheterocycles [13][14][15].…”

New Small-Molecule Synthetic Antimycobacterials

“…The leading compound in a series of 1,3-thiazine derivatives, compound 37 (Table 2), displays good antimycobacterial activity (55,56); no toxicity data were reported. These compounds have relatively low molecular weights and three potential points of diversity, making them attractive templates for high-throughput analogue synthesis.…”

Synthesis and antimicrobial activities of some thieno[3,2-d][1,3]thiazine nucleosides derivatives

“…5,6-Dihydro-4H-1,3-thiazines were synthesized as cholecystokinin antagonists [4] or antimycobacterial [5]. Heterocyclic compounds containing on the thiazine includes carbon and nitrogen atoms and one sulfur atom in different locations on the six-membered ring in there is 1,2-; 1,3-; 1,4-thiazines [6][7][8] and include derivatives were synthesized NCS binding to use antibacterial, antimicrobial, insects, anti-tumor, fungal, and agents herbicides, and various colorants etc.…”